SCHEMBL9157129

SCHEMBL9157129

COc1cccc(-c2ccccc2C(=O)NC(C)=O)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.62
KDM4E B2RXH2 2/20 0.62
HSP90AA1 P07900 2/20 0.53
HSP90AB1 P08238 2/20 0.53
CDK4 P11802 1/20 0.53
CCND1 P24385 1/20 0.53
POLB P06746 1/20 0.52
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
RAB9A P51151 2/20 0.49
ADORA3 P0DMS8 2/20 0.48
ADORA2B P29275 2/20 0.48
ADORA1 P30542 2/20 0.48
ADORA2A P29274 1/20 0.48
ALDH1A1 P00352 3/20 0.47
HSD17B10 Q99714 3/20 0.47
TSHR P16473 1/20 0.47
HTT P42858 2/20 0.47
NPC1 O15118 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL977594 0.86 GAA (0.65) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL9117254 0.84 GAA (0.63) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL1515816 0.84 GAA (0.62) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL30285198 0.82 SLC6A3 (0.66) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL8887143 0.82 GAA (0.59) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL6300807 0.81 GAA (0.80) GAAKDM4EPOLBRAB9AALDH1A1
SCHEMBL496484 0.81 KDM4E (0.62) GAAKDM4EPOLBRAB9AALDH1A1
SCHEMBL4709256 0.80 BCAT2 (0.59) GAAKDM4ECDK4CCND1RAB9A
SCHEMBL7894667 0.80 GAA (0.57) GAAKDM4EHSP90AA1HSP90AB1CDK4
SCHEMBL6295717 0.78 GAA (0.70) GAAKDM4EPOLBRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5410054-A Heteroaryl quinolines as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1995-04-25 US disclosed
WO-1995003300-A1 HETEROARYL QUINOLINES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1995-02-02 WO disclosed