SCHEMBL9158263

SCHEMBL9158263

CCc1ccc(-c2ccc(F)nc2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
CYP2A6 P11509 3/20 0.44
CYP2B6 P20813 3/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
GRIN1 Q05586 3/20 0.40
GRIN2B Q13224 3/20 0.40
FEN1 P39748 3/20 0.40
ALOX5AP P20292 2/20 0.40
USP7 Q93009 1/20 0.39
WNT3A P56704 2/20 0.38
RARB P10826 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
GRM5 P41594 1/20 0.38
CYP2E1 P05181 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9156736 0.94 PDE3B (0.42) PDE3BPDE3ACYP2A6CYP2B6CYP3A4
SCHEMBL9162226 0.88 NPC1 (0.45) PDE3BPDE3ACYP2A6CYP2B6CYP3A4
SCHEMBL9155798 0.85 RARB (0.49) PDE3BPDE3ACYP2A6CYP2B6CYP3A4
SCHEMBL9766599 0.85 RARB (0.50) PDE3BPDE3ARARB
SCHEMBL9152755 0.84 RARB (0.54) PDE3BPDE3ACYP2A6CYP2B6CYP3A4
SCHEMBL9155782 0.83 RARB (0.56) CYP3A4RARB
SCHEMBL9160685 0.83 RARB (0.56) CYP3A4RARB
SCHEMBL9154043 0.82 NPC1 (0.43) PDE3BPDE3ACYP2A6CYP2B6CYP3A4
SCHEMBL10981111 0.81 CHKA (0.45) CYP2A6RARB
SCHEMBL8774259 0.81 FEN1 (0.40) PDE3BPDE3AGRIN1GRIN2BFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
US-5205962-A Stable liquid crystals MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-04-27 US disclosed