SCHEMBL9159266

SCHEMBL9159266

CC1(C)CC(Cl)c2cc(C#N)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 7/20 0.40
PGR P06401 1/20 0.39
KDM1A O60341 2/20 0.38
CYP11B2 P19099 2/20 0.38
ABCC9 O60706 3/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.38
CHRNA1 P02708 1/20 0.37
CHRNG P07510 1/20 0.37
CHRNB1 P11230 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9160473 0.81 KDM1A (0.44) ABCB1PGRKDM1ACYP11B2ABCC9
SCHEMBL9158928 0.81 PGR (0.53) ABCB1PGRKDM1ACYP11B2ABCC9
SCHEMBL9032284 0.74 ABCB1 (0.46) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL25444478 0.71 KDM1A (0.48) ABCB1PGRKDM1ACYP11B2ABCC9
SCHEMBL10512412 0.71 PGR (0.60) ABCB1PGRKDM1ACYP11B2ABCC9
SCHEMBL11744995 0.70 HTR2C (0.38) CYP2D6CYP2C19
SCHEMBL16905203 0.68 PGR (0.42) ABCB1PGRKDM1ACYP11B2NSD2
SCHEMBL2223445 0.68 RARB (0.53) PGRKDM1ANSD2DRD2DRD3
SCHEMBL17771666 0.66 XIAP (0.46) ABCB1PGRNSD2DRD2DRD3
SCHEMBL24489941 0.65 ABCB1 (0.36) ABCB1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5401848-A Indane and quinoline derivatives E. R. SQUIBB & SONS, INC. (US) 1995-03-28 US disclosed
EP-0488616-A1 Indane and quinoline derivatives E.R. SQUIBB & SONS, INC. (US) 1992-06-03 EP disclosed