SCHEMBL9159435

SCHEMBL9159435

CCCCCCCCCCCCCCOc1ccc(CC(=O)Nc2ccc(-n3ccnc3C)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.62
CYP3A4 P08684 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP19A1 P11511 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
PORCN Q9H237 1/20 0.57
MAPT P10636 1/20 0.52
TP53 P04637 2/20 0.50
GAA P10253 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
PDE4A P27815 1/20 0.48
HIF1A Q16665 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ALDH1A1 P00352 1/20 0.46
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9168856 0.99 CYP2D6 (0.61) CYP2D6CYP3A4CYP1A2CYP19A1CYP2C9
SCHEMBL9625793 0.89 CYP2D6 (0.52) CYP2D6CYP3A4CYP1A2CYP19A1CYP2C9
Hydrochloric Acid SCHEMBL9625800 0.88 CYP2D6 (0.51) CYP2D6CYP3A4CYP1A2CYP19A1CYP2C9
Iodide SCHEMBL9166011 0.82 MAPT (0.47) CYP2D6CYP1A2CYP2C19MAPTGAA
Iodide SCHEMBL9166019 0.79 SMN1; SMN2 (0.49) CYP2D6CYP1A2MAPTGAAL3MBTL1
SCHEMBL9166917 0.78 SMN1; SMN2 (0.59) CYP2D6CYP1A2MAPTGAAL3MBTL1
Iodide SCHEMBL9166006 0.74 GAA (0.47) CYP2D6CYP1A2MAPTGAAL3MBTL1
Hydrochloric Acid SCHEMBL9167327 0.74 MAPT (0.48) CYP2D6CYP1A2MAPTGAAL3MBTL1
SCHEMBL10760230 0.73 CYP3A4 (0.57) CYP2D6CYP3A4CYP1A2CYP19A1CYP2C9
SCHEMBL16198332 0.73 PORCN (1.00) CYP2D6CYP3A4CYP1A2CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5432189-A Bis-aryl amide and urea antagonists of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1995-07-11 US disclosed
US-5350759-A Bis-aryl urea compounds WISSNER ALLAN (US) 1994-09-27 US disclosed
US-5231182-A Platelet activating factor inhibitor AMERICAN CYANAMID COMPANY (US) 1993-07-27 US disclosed
US-5225425-A Respiratory system disorders AMERICAN CYANAMID COMPANY (US) 1993-07-06 US disclosed
US-5128351-A BIS-ARYL AMIDE AND UREA ANTAGONISTS OF PLATELET ACTIVATING FACTOR AMERICAN CYANAMID COMPANY (US) 1992-07-07 US disclosed
US-5077409-A Reducing hydroxy bis-aryl amide, acylating, hydrolyzing, sulfonating, halogenating, alkylating with nitrogen heterocycle AMERICAN CYANAMID COMPANY (US) 1991-12-31 US disclosed
EP-0458037-A1 Bis-aryl amide and urea antagonists of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1991-11-27 EP disclosed