SCHEMBL9161994

SCHEMBL9161994

Nc1cnc2ccc(Cl)cc2c1-c1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.53
NPSR1 Q6W5P4 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAP4K4 O95819 3/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
STAT3 P40763 1/20 0.42
SOS2 Q07890 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9159565 0.91 HSP90AB1 (0.52) NR4A2NPSR1KDM4EMAP4K4ALDH1A1
SCHEMBL9161172 0.90 ALDH1A1 (0.52) NR4A2NPSR1KDM4EALDH1A1CYP3A4
Ammonia Solution, Strong SCHEMBL2249468 0.89 ALDH1A1 (0.51) NR4A2NPSR1KDM4EALDH1A1CYP3A4
SCHEMBL9164555 0.86 MAP4K4 (0.51) NR4A2NPSR1KDM4EMAP4K4ALDH1A1
SCHEMBL9164875 0.82 TSHR (0.56) NR4A2KDM4EALDH1A1CA12CA1
SCHEMBL18658904 0.79 NR4A2 (0.59) NR4A2MAP4K4ALDH1A1CYP3A4LMNA
SCHEMBL30155016 0.79 NR4A2 (0.59) NR4A2MAP4K4ALDH1A1CYP3A4LMNA
SCHEMBL8835043 0.78 NR4A2 (0.47) NR4A2NPSR1KDM4EALDH1A1CYP3A4
SCHEMBL28458986 0.77 NR4A2 (0.58) NR4A2ALDH1A1CYP3A4LMNACYP1A2
Ammonia Solution, Strong SCHEMBL2251166 0.77 GRM5 (0.50) NR4A2SOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 EP disclosed
US-5254565-A Enzyme inhibitors; anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-19 US disclosed
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed