SCHEMBL9164875

SCHEMBL9164875

COc1ccc(-c2c(N)cnc3ccc(Cl)cc23)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.56
MAPK1 P28482 1/20 0.56
CASP1 P29466 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
KIT P10721 2/20 0.43
NR4A2 P43354 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 2/20 0.42
FYN P06241 1/20 0.42
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
MTOR P42345 1/20 0.41
PIK3CG P48736 1/20 0.41
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9161994 0.82 NR4A2 (0.53) CA1CA2NR4A2ALDH1A1KDM4E
SCHEMBL9090774 0.80 AMY1A (0.44) TSHRMAPK1CASP1HSD17B10NR4A2
SCHEMBL9163823 0.80 SMN1; SMN2 (0.51) TSHRMAPK1CASP1HSD17B10CA1
SCHEMBL9159565 0.80 HSP90AB1 (0.52) NR4A2ALDH1A1KDM4EMAPT
SCHEMBL9162830 0.80 MAP2 (0.47) TSHRMAPK1HSD17B10PDGFRBPDGFRA
SCHEMBL9164555 0.78 MAP4K4 (0.51) NR4A2ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9159337 0.77 LMNA (0.43) TSHRMAPK1CASP1HSD17B10NR4A2
SCHEMBL9161172 0.76 ALDH1A1 (0.52) MAPK1NR4A2ALDH1A1KDM4EHPGD
Ammonia Solution, Strong SCHEMBL2249468 0.75 ALDH1A1 (0.51) MAPK1NR4A2ALDH1A1KDM4EHPGD
SCHEMBL25493265 0.74 NR4A2 (0.42) KITNR4A2ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-B1 Quinoline derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-01-25 EP disclosed
US-5254565-A Enzyme inhibitors; anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-19 US disclosed
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed