SCHEMBL9163000

SCHEMBL9163000

CC(C)(C=O)Oc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
CHRNB2 P17787 5/20 0.41
CHRNA4 P43681 5/20 0.41
ALDH1A1 P00352 1/20 0.41
THRB P10828 1/20 0.41
KMT2A Q03164 1/20 0.40
KIF11 P52732 1/20 0.40
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
GALR3 O60755 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
HTT P42858 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2732089 0.79 LMNA (0.50) LMNATDP1CHRNB2CHRNA4KMT2A
SCHEMBL29583666 0.79 LMNA (0.50) LMNATDP1CHRNB2CHRNA4KMT2A
SCHEMBL2401039 0.79 LMNA (0.43) LMNATDP1CHRNB2CHRNA4KMT2A
SCHEMBL27983764 0.77 CHRNB2 (0.50) LMNATDP1CHRNB2CHRNA4CYP11B1
SCHEMBL6210928 0.77 CA4 (0.39) LMNATDP1ALDH1A1KMT2AMAPK1
SCHEMBL3372165 0.74 PPARA (0.50) ALDH1A1THRBKMT2A
SCHEMBL26146529 0.73 LMNA (0.44) LMNATDP1CHRNB2CHRNA4KMT2A
SCHEMBL28206059 0.72 KMT2A (0.54) LMNATDP1CHRNB2CHRNA4ALDH1A1
SCHEMBL7099252 0.71 CHRNB2 (0.45) LMNATDP1CHRNB2CHRNA4CYP11B1
SCHEMBL130691 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040753-C Pyridine derivatives and the preparation thereof ICI PLC (GB) 1998-11-18 CN disclosed
US-5401849-A FOR ANTAGONIZING THE ACTIONS OF, AND INHIBITING THE SYNTHESIS OF, THROMBOXANE A2 ZENECA LIMITED (GB) 1995-03-28 US disclosed
EP-0329360-B1 Pyridine derivatives ICI PLC (GB) 1994-08-03 EP disclosed
US-5248780-A Thromboxane inhibitors IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1993-09-28 US disclosed
US-5166213-A Antiischemic agents, cardiovascular disorders, antiasthmatics or antiinflammatory agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
EP-0288279-B1 1,3-DIOXANES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-09-09 EP disclosed
CN-1015893-B 1,3-DIOXANES ICI LTD (GB) 1992-03-18 CN disclosed
US-4921866-A 1,3-dioxanes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-05-01 US disclosed
CN-1035115-A Pyridine derivate and preparation method thereof ICI PLC (GB) 1989-08-30 CN disclosed
EP-0329360-A2 Pyridine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-08-23 EP disclosed
CN-88102356-A 1,3-two  alkanes 1988-12-28 CN disclosed
EP-0288279-A2 1,3-Dioxanes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-10-26 EP disclosed