SCHEMBL9164075

SCHEMBL9164075

O=C(NCc1ccccc1)c1cc([N+](=O)[O-])ccc1O

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.60
KMT2A Q03164 5/20 0.60
GAA P10253 1/20 0.59
MAPT P10636 1/20 0.59
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
HPGD P15428 1/20 0.56
CYP2C19 P33261 1/20 0.56
CTSB P07858 1/20 0.56
HSP90AA1 P07900 1/20 0.56
AKR1C3 P42330 1/20 0.53
KCNMA1 Q12791 1/20 0.53
SYK P43405 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
TUBB P07437 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940724 0.88 MEN1 (0.61) MEN1KMT2AGAAMAPTCYP1A2
SCHEMBL28763268 0.87 NPC1 (0.66) MEN1KMT2AMAPTCYP1A2HPGD
SCHEMBL9162776 0.85 MEN1 (0.54) MEN1KMT2AGAAMAPTCYP1A2
SCHEMBL6944295 0.85 MEN1 (0.58) MEN1KMT2AGAAMAPTCYP1A2
SCHEMBL9162780 0.85 MEN1 (0.58) MEN1KMT2AGAAMAPTCYP1A2
SCHEMBL16043211 0.83 ALDH1A1 (0.58) MEN1KMT2AMAPTHPGDKCNMA1
SCHEMBL26098852 0.82 CYP1A2 (0.63) MEN1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL9162784 0.81 HSP90AA1 (0.52) MEN1KMT2AGAACYP1A2CYP3A4
SCHEMBL13753896 0.80 L3MBTL1 (0.57) MEN1KMT2AGAAMAPTCYP1A2
SCHEMBL13385655 0.80 MEN1 (0.63) MEN1KMT2AMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641311-A1 NOVEL DIHYDROXYBENZYLAMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Aventis Pharma S.A. (FR) 1995-03-08 EP disclosed
WO-1993023364-A1 NOVEL DIHYDROXYBENZYLAMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1993-11-25 WO disclosed