SCHEMBL9165115

SCHEMBL9165115

CCCCCCCCc1ccc(-c2ncc(O)cn2)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.50
PTGS2 P35354 4/20 0.47
ESR1 P03372 2/20 0.47
ADRA2A P08913 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
TACR2 P21452 2/20 0.47
SLC6A2 P23975 2/20 0.47
SLC6A4 P31645 2/20 0.47
SLC6A3 Q01959 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP3A4 P08684 2/20 0.47
LMNA P02545 1/20 0.47
SHBG P04278 1/20 0.47
TP53 P04637 1/20 0.47
HSPD1 P10809 1/20 0.47
ADRB3 P13945 1/20 0.47
HTR2C P28335 1/20 0.47
HSPE1 P61604 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9399034 0.90 RARB (0.50) RARBPTGS2ESR1ADRA2AADORA3
SCHEMBL9399411 0.89 RARB (0.48) RARBESR1ADRA2AADORA3TACR2
SCHEMBL8555801 0.86 RAB9A (0.49) RARBPTGS2ESR1ADRA2AADORA3
SCHEMBL9399921 0.86 RARB (0.52) RARBKDM4EALDH1A1HSD17B10TP53
SCHEMBL9398829 0.86 RARB (0.46) RARBKDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL9398666 0.86 RARB (0.49) RARBPTGS2ESR1ADRA2AADORA3
SCHEMBL8992409 0.84 RAB9A (0.56) RARBPTGS2ESR1ADRA2AADORA3
SCHEMBL9449622 0.84 RAB9A (0.56) RARBPTGS2ESR1ADRA2AADORA3
SCHEMBL9399018 0.84 RARB (0.53) RARBKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8984207 0.84 RARB (0.54) RARBPTGS2ESR1ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0428665-B1 FLUOROPHENYL PYRIMIDINES MERCK PATENT GMBH (DE) 1995-04-05 EP disclosed
US-5340497-A Ferroelectric liquid crystal MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-08-23 US disclosed
EP-0428665-A1 FLUOROPHENYL PYRIMIDINES. MERCK PATENT GMBH (DE) 1991-05-29 EP disclosed
WO-1990015116-A1 FLUOROPHENYL PYRIMIDINES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-12-13 WO disclosed