SCHEMBL9166247

SCHEMBL9166247

N#CC(C(=O)Nc1cccc(Cl)c1)C(=O)c1nn(-c2ccccc2)c2c1Cc1ccc(C(=O)O)cc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.40
KCNJ6 P48051 4/20 0.38
KCNJ3 P48549 4/20 0.38
KCNJ5 P48544 3/20 0.38
MAPT P10636 4/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
IKBKB O14920 1/20 0.36
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
TP53 P04637 1/20 0.35
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171534 0.93 IKBKB (0.34) ALDH1A1IKBKBCCNA2CDK2CCNA1
SCHEMBL9175603 0.91 IKBKB (0.41) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9174817 0.91 RIPK1 (0.43) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9171500 0.91 RIPK1 (0.40) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9174674 0.91 RIPK1 (0.44) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9176550 0.90 KMT2A (0.43) RIPK1MAPTALDH1A1KDM4EHSD17B10
SCHEMBL9174505 0.89 IKBKB (0.39) RIPK1ALDH1A1IKBKBLMNA
SCHEMBL9174664 0.89 IDO1 (0.44) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9837095 0.89 RIPK1 (0.39) RIPK1KCNJ6KCNJ3KCNJ5MAPT
SCHEMBL9836709 0.88 IKBKB (0.41) RIPK1KCNJ6KCNJ3KCNJ5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424308-A Immunomodulating agents FARMITALIA CARLO ERBA S.R.L. (IT) 1995-06-13 US disclosed
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed