SCHEMBL9836709

SCHEMBL9836709

N#CC(C(=O)Nc1ccc(F)cc1)C(=O)c1nn(-c2ccccc2)c2c1Cc1ccc(C(=O)O)cc1-2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 13/20 0.41
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
RIPK1 Q13546 1/20 0.39
KCNJ6 P48051 1/20 0.37
KCNJ5 P48544 1/20 0.37
KCNJ3 P48549 1/20 0.37
P2RY1 P47900 1/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
CHUK O15111 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R2 O00459 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3R5 Q8WYR1 1/20 0.35
PIK3R3 Q92569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171534 0.95 IKBKB (0.34) IKBKBALDH1A1MEN1KMT2APIK3CD
SCHEMBL9167969 0.93 IKBKB (0.43) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL9172382 0.91 IKBKB (0.42) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL8132620 0.91 IKBKB (0.40) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL9171221 0.90 RIPK1 (0.43) IKBKBALDH1A1LMNARIPK1P2RY1
SCHEMBL9173723 0.90 IKBKB (0.44) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL9173066 0.90 ALDH1A1 (0.41) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL9170158 0.89 ALDH1A1 (0.42) IKBKBALDH1A1RIPK1P2RY1MEN1
SCHEMBL9174751 0.89 IKBKB (0.41) IKBKBALDH1A1LMNARIPK1KCNJ6
SCHEMBL9173782 0.88 MAPK14 (0.42) IKBKBALDH1A1LMNARIPK1P2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422051-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-04-17 EP disclosed
WO-1989012630-A1 CONDENSED PYRAZOLE 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed
EP-0347773-A1 Condensed Pyrazole 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1989-12-27 EP disclosed