SCHEMBL9176240

SCHEMBL9176240

N[C@@H](CCSc1ncnc2[nH]cnc12)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.39
SLC6A5 Q9Y345 1/20 0.36
IDO1 P14902 1/20 0.35
CYP3A4 P08684 1/20 0.35
SLC7A5 Q01650 1/20 0.35
BHMT Q93088 2/20 0.34
TSHR P16473 1/20 0.34
DOT1L Q8TEK3 4/20 0.34
CARM1 Q86X55 2/20 0.34
EHMT2 Q96KQ7 2/20 0.34
DNMT1 P26358 2/20 0.34
PRMT1 Q99873 2/20 0.34
DNMT3B Q9UBC3 2/20 0.34
TRDMT1 O14717 1/20 0.34
PRMT5 O14744 1/20 0.34
SUV39H1 O43463 1/20 0.34
PRMT3 O60678 1/20 0.34
INMT O95050 1/20 0.34
NSD2 O96028 1/20 0.34
PNMT P11086 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9176272 1.00 NOTUM (0.39) NOTUMSLC6A5IDO1CYP3A4SLC7A5
SCHEMBL9177267 0.86 NOTUM (0.41) NOTUMSLC6A5CYP3A4SLC7A5TSHR
SCHEMBL13401493 0.81 SLC6A5 (0.47) NOTUMSLC6A5TSHR
SCHEMBL30999504 0.81 TSHR (0.56) TSHR
SCHEMBL9176257 0.81 TSHR (0.56) TSHR
SCHEMBL9176248 0.81 TSHR (0.56) TSHR
SCHEMBL735449 0.79 NOTUM (0.60) NOTUMTSHRKMT2A
Adenine SCHEMBL9663399 0.79 MARS1 (0.43) DOT1LCARM1EHMT2DNMT1PRMT1
SCHEMBL14347081 0.78 SLC6A5 (0.54) NOTUMSLC6A5TSHR
Adenine SCHEMBL23928076 0.78 MARS1 (0.42) TSHRDOT1LCARM1EHMT2DNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426467-B1 Prodrugs of 6-mercaptopurine and 6-thioguanine WISCONSIN ALUMNI RES FOUND (US) 1995-04-05 EP disclosed
US-5120740-A PRODRUGS OF 6-MERCAPTOPURINE AND 6-THIOGUANINE WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1992-06-09 US disclosed
EP-0426467-A1 Prodrugs of 6-mercaptopurine and 6-thioguanine WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1991-05-08 EP disclosed