SCHEMBL9178259

SCHEMBL9178259

O=C(O)c1ccccc1C(=O)c1ccccc1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.61
ALOX15 P16050 3/20 0.61
AKR1C3 P42330 3/20 0.59
CES2 O00748 1/20 0.58
CES1 P23141 1/20 0.58
ALB P02768 1/20 0.55
CDC25B P30305 3/20 0.55
CDC25A P30304 1/20 0.52
HSD17B10 Q99714 1/20 0.52
ATM Q13315 1/20 0.52
KMT2A Q03164 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
PRNP P04156 1/20 0.50
NR4A1 P22736 1/20 0.50
PTPN1 P18031 1/20 0.48
ERCC5 P28715 1/20 0.48
FEN1 P39748 1/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27185988 0.91 CES2 (0.68) ALDH1A1ALOX15CES2CES1ALB
SCHEMBL31574193 0.91 CES2 (0.68) ALDH1A1ALOX15CES2CES1ALB
SCHEMBL30293901 0.89 CES2 (0.71) ALDH1A1ALOX15CES2CES1ALB
SCHEMBL250099 0.89 CES2 (0.71) ALDH1A1ALOX15CES2CES1ALB
SCHEMBL29362443 0.86 CES2 (0.68) ALDH1A1ALOX15AKR1C3CES2CES1
SCHEMBL97828 0.86 CES2 (0.68) ALDH1A1ALOX15AKR1C3CES2CES1
SCHEMBL30968201 0.86 CES2 (0.68) ALDH1A1ALOX15AKR1C3CES2CES1
Hydrochloric Acid SCHEMBL27733532 0.86 CES2 (0.68) ALDH1A1ALOX15CES2CES1ALB
SCHEMBL29977835 0.86 ALDH1A1 (0.82) ALDH1A1ALOX15AKR1C3CDC25BCDC25A
SCHEMBL11402284 0.86 ALDH1A1 (0.82) ALDH1A1ALOX15AKR1C3CDC25BCDC25A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481383-B1 Heterocyclic amine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-06-28 EP disclosed
US-5300646-A Intermediates for acylcoenzyme A:cholesterol acyltransferase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-05 US disclosed
US-5198462-A Acyl Coenzyme A:Cholesterol Transferase Inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-03-30 US disclosed
EP-0481383-A1 Heterocyclic amine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-22 EP disclosed
US-4505921-A Sulfonylurea compounds and their use in treating diabetes ADIR, S.A.R.L. (FR) 1985-03-19 US disclosed