SCHEMBL9178289

SCHEMBL9178289

CC(C)N1CCC(Sc2c[nH]c3ccc(Cl)cc23)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 8/20 0.45
TUBB4A P04350 3/20 0.45
TUBB P07437 3/20 0.45
TUBA3C P0DPH7 3/20 0.45
TUBA1B P68363 3/20 0.45
TUBA4A P68366 3/20 0.45
TUBB4B P68371 3/20 0.45
TUBB3 Q13509 3/20 0.45
TUBB2A Q13885 3/20 0.45
TUBB8 Q3ZCM7 3/20 0.45
TUBA3E Q6PEY2 3/20 0.45
TUBA1A Q71U36 3/20 0.45
TUBA1C Q9BQE3 3/20 0.45
TUBB6 Q9BUF5 3/20 0.45
TUBB2B Q9BVA1 3/20 0.45
TUBB1 Q9H4B7 3/20 0.45
HTR2A P28223 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171444 0.86 IDO1 (0.48) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9176461 0.85 IDO1 (0.42) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9177126 0.83 IDO1 (0.48) IDO1TUBB4ATUBBTUBA3CTUBA1B
Hydrochloric Acid SCHEMBL9176166 0.82 OPRM1 (0.46) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9038781 0.80 F7 (0.47) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9178079 0.79 SLC6A4 (0.53) IDO1TUBB4ATUBBTUBA3CTUBA1B
Hydrochloric Acid SCHEMBL9176359 0.78 SLC6A4 (0.52) IDO1TUBB4ATUBBTUBA3CTUBA1B
Hydrochloric Acid SCHEMBL9171641 0.77 OPRM1 (0.65) IDO1OPRM1OPRK1OPRL1SLC6A4
SCHEMBL9173510 0.74 HTR1D (0.49) HTR2A
SCHEMBL9176103 0.74 F7 (0.38) IDO1TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5418242-A Piperidinylthioindole derivatives, their methods of preparation and pharmaceutical compositions in which they are present, useful especially as analgesics LABORATOIRES UPSA (FR) 1995-05-23 US disclosed
US-5317025-A Piperidinylthioindole derivatives, their methods of preparation and pharmaceutical compositions in which they are present, useful especially as analgesics LABORATOIRES USPA (FR) 1994-05-31 US disclosed