SCHEMBL9178367

SCHEMBL9178367

c1ccc2c(c1)CC(CCN1CCN(c3cccc4c3OCCO4)CC1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.64
LMNA P02545 1/20 0.64
CYP3A4 P08684 1/20 0.64
HTR1A P08908 1/20 0.64
ALOX12 P18054 1/20 0.64
MAPK1 P28482 1/20 0.64
PMP22 Q01453 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9175474 0.93 HTR1A (0.65) HTR1A
SCHEMBL9179406 0.88 HTR1A (0.67) ALDH1A1LMNACYP3A4HTR1AALOX12
SCHEMBL1037297 0.85
SCHEMBL1038535 0.82
SCHEMBL9183299 0.81 HTR1A (0.58) ALDH1A1LMNACYP3A4HTR1AALOX12
SCHEMBL9176472 0.81
SCHEMBL9180759 0.80 HTR1A (0.63) HTR1A
SCHEMBL6173953 0.79 HTR1A (0.65) HTR1A
SCHEMBL8688384 0.79 HTR1A (0.65) HTR1A
SCHEMBL31051744 0.79 HTR1A (0.65) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490772-B1 1,4-Disubstituted piperazines, their process of preparation and pharmaceutical compositions containing them ADIR (FR) 1995-07-26 EP disclosed
US-5194437-A Substituted with oxygen containing heterocycle, central nervous system disorders, neuroendocrine disorders ADIR ET COMPAGNIE (FR) 1993-03-16 US disclosed
EP-0490772-A1 1,4-Disubstituted piperazines, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-06-17 EP disclosed