SCHEMBL9178705

SCHEMBL9178705

O=C(Nc1ccc(F)cc1F)Nc1oc(=O)c2ccccc2c1-c1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.51
RAB9A P51151 3/20 0.51
NPC1 O15118 2/20 0.51
HTT P42858 2/20 0.51
POLB P06746 2/20 0.51
MAPT P10636 3/20 0.50
PKM P14618 1/20 0.50
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 2/20 0.49
RECQL P46063 2/20 0.46
GAA P10253 2/20 0.44
TP53 P04637 1/20 0.44
PTGS2 P35354 1/20 0.44
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 1/20 0.43
KLK7 P49862 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9174188 0.95 POLB (0.56) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9179564 0.92 RAB9A (0.46) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9175479 0.87 MAPT (0.45) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9182119 0.85 POLB (0.58) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9175907 0.85 POLB (0.58) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9178041 0.83 NPC1 (0.53) SMN1; SMN2RAB9ANPC1HTTMAPT
SCHEMBL9178393 0.78 TACR1 (0.57) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL27193044 0.72 RAB9A (0.77) SMN1; SMN2RAB9ANPC1HTTPOLB
SCHEMBL9260108 0.70 SMN1; SMN2 (0.48) SMN1; SMN2RAB9ANPC1HTTMAPT
SCHEMBL9278296 0.70 POLB (0.52) SMN1; SMN2RAB9ANPC1HTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481383-B1 Heterocyclic amine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-06-28 EP disclosed
US-5300646-A Intermediates for acylcoenzyme A:cholesterol acyltransferase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-05 US disclosed
US-5198462-A Acyl Coenzyme A:Cholesterol Transferase Inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-03-30 US disclosed
EP-0481383-A1 Heterocyclic amine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-22 EP disclosed