SCHEMBL9185482

SCHEMBL9185482

CCOC(=O)c1[nH]c2ccc(OC)cc2c1CC(=O)O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.71
KDM4E B2RXH2 6/20 0.71
HPGD P15428 5/20 0.71
MAPT P10636 3/20 0.71
NPC1 O15118 1/20 0.71
RAB9A P51151 1/20 0.71
AKR1C2 P52895 1/20 0.69
NQO2 P16083 1/20 0.67
HSD17B10 Q99714 5/20 0.63
LMNA P02545 3/20 0.63
HTT P42858 1/20 0.63
PTGS1 P23219 1/20 0.62
PTGS2 P35354 1/20 0.62
TUBB4A P04350 3/20 0.58
TUBB P07437 3/20 0.58
TUBA3C P0DPH7 3/20 0.58
TUBA1B P68363 3/20 0.58
TUBA4A P68366 3/20 0.58
TUBB4B P68371 3/20 0.58
TUBB3 Q13509 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958468 0.90 ALDH1A1 (0.71) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL29628777 0.90 ALDH1A1 (0.71) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL29198788 0.86 KDM4E (0.66) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL29628842 0.86 KDM4E (0.76) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL27566660 0.84 NQO2 (0.72) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL6353272 0.84 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9189433 0.84 ALDH1A1 (0.65) ALDH1A1KDM4EHPGDMAPTTUBB4A
SCHEMBL7511884 0.84 DRD2 (0.61) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL3954004 0.83 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL3993248 0.83 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0394905-B1 Excitatory amino acid antagonists MERRELL DOW PHARMA (US) 1995-08-16 EP claimed
EP-0394905-B1 Excitatory amino acid antagonists MERRELL DOW PHARMA (US) 1995-08-16 EP disclosed