SCHEMBL9186142

SCHEMBL9186142

Cc1ccc(S(=O)(=O)N(CCCN)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.58
CA12 O43570 1/20 0.54
CA9 Q16790 1/20 0.54
KMT2A Q03164 3/20 0.53
CNR2 P34972 3/20 0.53
CNR1 P21554 2/20 0.53
MEN1 O00255 1/20 0.53
KEAP1 Q14145 1/20 0.52
NFE2L2 Q16236 1/20 0.52
LMNA P02545 2/20 0.50
NR3C1 P04150 1/20 0.50
MAPT P10636 1/20 0.50
ALDH1A1 P00352 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
BACE1 P56817 1/20 0.48
BMP1 P13497 1/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8466425 0.87 ESR1 (0.76) ESR1CA12CA9KMT2ACNR2
SCHEMBL9188513 0.84 ESR1 (0.57) ESR1CA12CA9KMT2ACNR2
SCHEMBL8224221 0.83 ESR1 (0.75) ESR1CA12CA9KMT2ACNR2
SCHEMBL28029865 0.82 CA12 (0.57) ESR1CA12CA9KMT2ACNR2
SCHEMBL9189756 0.82 ESR1 (0.54) ESR1CA12CA9KMT2ACNR2
SCHEMBL14502622 0.81 KEAP1 (0.66) ESR1CA12CA9KMT2ACNR2
SCHEMBL9702124 0.81 CNR2 (0.65) ESR1CA12CA9KMT2ACNR2
SCHEMBL6204172 0.80 ESR1 (0.55) ESR1KMT2ACNR2CNR1MEN1
SCHEMBL9184943 0.80 ESR1 (0.52) ESR1CA12CA9KMT2ACNR2
SCHEMBL28245407 0.80 ESR1 (0.55) ESR1CA12CA9KMT2ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497202-B1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMA (US) 1995-09-13 EP disclosed
US-5217964-A POLYAMINE THIOLS AS RADIOPROTECTIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US disclosed
EP-0497202-A1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-08-05 EP disclosed