SCHEMBL9192568

SCHEMBL9192568

CC1CCN(Cc2ccc(CC#N)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.67
ACHE P22303 5/20 0.62
HTR7 P34969 4/20 0.48
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 1/20 0.43
KCNA3 P22001 1/20 0.41
NCF1 P14598 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14375216 0.83 HRH3 (0.67) HRH3ACHE
SCHEMBL3440098 0.80 HRH3 (0.65) HRH3ALDH1A1KDM4ESMN1; SMN2NCF1
SCHEMBL3594477 0.79 LMNA (0.61) HRH3ALDH1A1KDM4ENCF1
SCHEMBL156202 0.79 HRH3 (0.76) HRH3ACHEALDH1A1KDM4E
SCHEMBL8252094 0.79 HRH3 (0.76) HRH3ACHEHTR7ALDH1A1KDM4E
SCHEMBL4010533 0.79 HRH3 (0.69) HRH3ALDH1A1KDM4ESMN1; SMN2NCF1
SCHEMBL8275450 0.79 HRH3 (0.76) HRH3ACHEALDH1A1
SCHEMBL6227268 0.78 MEN1 (0.68) KCNA3
SCHEMBL3861163 0.77 HRH3 (0.73) HRH3ACHEHTR7ALDH1A1PARP1
SCHEMBL3004249 0.77 HRH3 (0.73) HRH3ACHEHTR7ALDH1A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0393534-B1 Pharmaceutically active pteridine derivatives ROEHM GMBH (DE) 1995-07-12 EP disclosed
US-5124326-A Antiarrhythmic, hypotensive agents; diuretics ROEHM GMBH CHEMISCHE FABRIK (DE) 1992-06-23 US disclosed
EP-0393534-A2 Pharmaceutically active pteridine derivatives RÖHM GMBH (DE) 1990-10-24 EP disclosed