SCHEMBL9192573

SCHEMBL9192573

COC(OC)c1cc(-c2ccccc2C=O)ccc1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPT P10636 2/20 0.40
CYP3A4 P08684 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
PRKDC P78527 1/20 0.40
ERN1 O75460 7/20 0.38
CYP19A1 P11511 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
STAT6 P42226 1/20 0.35
HIF1A Q16665 1/20 0.35
PHLPP2 Q6ZVD8 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4273991 0.73 VCAM1 (0.54) ALDH1A1MAPTERN1
SCHEMBL9664960 0.73 TDP1 (0.60) ALDH1A1MAPTCYP3A4ALOX15ERN1
SCHEMBL9730400 0.73 ALDH1A1 (0.50) ALDH1A1CYP3A4HSD17B10ERN1TP53
SCHEMBL9798217 0.73 ERN1 (0.43) ALDH1A1ERN1TDP1
SCHEMBL7383362 0.71 ALDH1A1 (0.60) ALDH1A1MAPTHSD17B10NPSR1CYP1A2
SCHEMBL2556452 0.71 ERN1 (0.50) ALDH1A1MAPTERN1TDP1
SCHEMBL10478265 0.70 HSD17B10 (0.46) ALDH1A1MAPTCYP3A4HSD17B10KDM4E
SCHEMBL3362982 0.69 ALDH1A1 (0.43) ALDH1A1MAPTKDM4ETDP1
SCHEMBL2928829 0.69 MAPK1 (0.53) ALDH1A1MAPTNPSR1MAPK1TDP1
SCHEMBL11287458 0.69 TDP1 (0.53) ALDH1A1MAPTCYP3A4MAPK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371564-B1 (1H-azol-1-ylmethyl)substituted quinoline, quinazoline or quinoxaline derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-07-12 EP disclosed
US-5037829-A Antitumor Activity; Androgen, Estrogen Inhibitors; Suppress The Plasma Elimination Of Retinoids JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-06 US disclosed
EP-0371564-A2 (1H-azol-1-ylmethyl)substituted quinoline, quinazoline or quinoxaline derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1990-06-06 EP disclosed