SCHEMBL9195181

SCHEMBL9195181

CCC(=O)c1cnc(N)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
KMT2A Q03164 2/20 0.46
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
BRAF P15056 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GSK3B P49841 1/20 0.33
MEN1 O00255 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9197924 0.86 MAPT (0.35) KMT2ANCOA1NCOA3KDM4ESMN1; SMN2
SCHEMBL9193763 0.81 MEN1 (0.36) HTTKMT2ANCOA1NCOA3KDM4E
SCHEMBL441934 0.80 HTT (0.50) HTTKMT2AHDAC1HDAC6SMN1; SMN2
SCHEMBL9197903 0.79 ALDH1A1 (0.43) HTTKMT2AMAPTALDH1A1
SCHEMBL9193384 0.79 CYP2D6 (0.45) HTTKDM4EALDH1A1GABRPGABRD
SCHEMBL451366 0.79 CYP2C19 (0.50) HTTKMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL8806697 0.79 HTT (0.48) HTTKMT2AHDAC1HDAC6KDM4E
SCHEMBL31276895 0.78 KMT2A (0.52) HTTKMT2AHDAC1HDAC6KDM4E
SCHEMBL7599288 0.78 KMT2A (0.52) HTTKMT2AHDAC1HDAC6KDM4E
SCHEMBL5904298 0.78 HTT (0.52) HTTKMT2ANCOA1NCOA3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299277-B1 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1995-10-18 EP disclosed
US-4990620-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1991-02-05 US disclosed
US-4927938-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1990-05-22 US disclosed
EP-0299277-A2 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1989-01-18 EP disclosed