SCHEMBL9195666

SCHEMBL9195666

COc1ccc(C(CCN(C)C)Oc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.78
HRH3 Q9Y5N1 5/20 0.78
SLC6A9 P48067 9/20 0.68
SLC6A2 P23975 2/20 0.52
SLC6A3 Q01959 2/20 0.52
KCNK2 O95069 1/20 0.52
KCNH2 Q12809 1/20 0.52
CACNA1C Q13936 1/20 0.52
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
TP53 P04637 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPK1 P28482 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17549671 0.89 SLC6A4 (0.78) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL679320 0.88 SLC6A4 (1.00) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL29700710 0.88 SLC6A4 (1.00) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL9197766 0.85 SLC6A4 (0.71) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL8971668 0.83 SLC6A4 (0.69) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
Oxalic Acid SCHEMBL4740319 0.83 SLC6A4 (0.72) SLC6A4HRH3SLC6A9CYP2D6CYP2C9
Oxalic Acid SCHEMBL7317614 0.82 SLC6A4 (0.88) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL5270870 0.81 SLC6A4 (0.70) SLC6A4HRH3SLC6A9SLC6A2
SCHEMBL7433161 0.81 SLC6A4 (0.69) SLC6A4HRH3SLC6A9SLC6A2SLC6A3
SCHEMBL17278117 0.80 SLC7A5 (0.76) SLC6A4HRH3SLC6A9SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399504-B1 Aryloxyphenylpropylamines their preparation and use NOVO NORDISK AS (DK) 1995-05-03 EP disclosed
US-5310756-A Aryloxyphenylpropylamines and their calcium overload blocking compositions and methods of use NOVO NORDISK A/S (DK) 1994-05-10 US disclosed
US-5145870-A Treating calcium overload in brain cells, anoxia, migraine, ischemia, epilepsy, neurodegenerative diseases NOVO NORDISK A/S (DK) 1992-09-08 US disclosed
EP-0399504-A2 Aryloxyphenylpropylamines their preparation and use NOVO NORDISK A/S (DK) 1990-11-28 EP disclosed