SCHEMBL9196642

SCHEMBL9196642

N=C(S)NCCCc1ccc(CSC(=N)N)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.56
IDO1 P14902 16/20 0.49
NPC1 O15118 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
RAB9A P51151 1/20 0.47
HIF1A Q16665 1/20 0.47
NOS3 P29474 1/20 0.47
NOS2 P35228 1/20 0.47
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5450413 0.75 NOS1 (1.00) NOS1IDO1NOS3NOS2
SCHEMBL9196649 0.75 NOS1 (0.56) NOS1IDO1NPC1CYP3A4CYP2D6
SCHEMBL14914554 0.73 ST14 (0.47) IDO1NPC1CYP2D6RAB9A
SCHEMBL14467311 0.73 HDAC1 (0.48) IDO1
SCHEMBL23116506 0.71 MAOB (0.47) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL18296627 0.67 ST14 (0.58)
SCHEMBL29074409 0.67 NPC1 (0.50) IDO1NPC1RAB9A
SCHEMBL23116515 0.67 MAOB (0.50) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL3779731 0.66 IDO1 (1.00) NOS1IDO1NOS3NOS2
SCHEMBL9198797 0.66 IDO1 (1.00) NOS1IDO1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670720-A1 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-09-13 EP disclosed
WO-1994012165-A2 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-06-09 WO disclosed