SCHEMBL9196836

SCHEMBL9196836

COC(=O)Oc1ccc(C(=O)N2CCN(CCc3ccccc3)CC2)nc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.56
PRKAA2 P54646 3/20 0.56
POLB P06746 1/20 0.53
GAA P10253 1/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
KCNH2 Q12809 1/20 0.52
PRKAB2 O43741 2/20 0.51
PRKAG1 P54619 2/20 0.51
PRKAA1 Q13131 2/20 0.51
PRKAG3 Q9UGI9 2/20 0.51
PRKAG2 Q9UGJ0 2/20 0.51
PRKAB1 Q9Y478 2/20 0.51
HTR2A P28223 1/20 0.47
LMNA P02545 1/20 0.46
THRB P10828 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SIGMAR1 Q99720 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9345715 0.83 PRKAA2 (0.66) DRD3PRKAA2POLBGAAMEN1
SCHEMBL517897 0.80 PRKAA2 (0.80) PRKAA2POLBGAAMEN1KMT2A
SCHEMBL15302927 0.78 PRKAA2 (0.61) PRKAA2POLBGAAMEN1KMT2A
SCHEMBL518286 0.77 PRKAA2 (0.69) PRKAA2MEN1KMT2AKCNH2PRKAB2
SCHEMBL518526 0.74 PRKAA2 (0.71) PRKAA2MEN1KMT2AKCNH2PRKAB2
SCHEMBL25284686 0.74 DRD2 (0.75) DRD3POLBGAAMEN1KMT2A
SCHEMBL25239004 0.72 PKM (0.78) DRD3GAAMEN1KMT2AKCNH2
SCHEMBL10284370 0.72 PRKAA2 (0.59) PRKAA2POLBGAAMEN1KMT2A
SCHEMBL9197096 0.72 P4HTM (0.53) POLBMEN1KMT2ALMNASMN1; SMN2
SCHEMBL9200180 0.72 HPGD (0.52) PRKAA2POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278452-B1 2,4- and 2,5-Pyridine-dicarboxylic-acid derivatives, process for their preparation, their use and medicines based on these compounds HOECHST AG (DE) 1995-05-24 EP disclosed