SCHEMBL9198063

SCHEMBL9198063

COc1ccc(CSC2C[C@@H](C(N)=O)N=C2N(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
EPHX1 P07099 1/20 0.38
FFAR1 O14842 1/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
MAPT P10636 2/20 0.35
LTA4H P09960 1/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204340 0.89 FFAR1 (0.37) IDO1FFAR1ALDH1A1HPGDSMN1; SMN2
SCHEMBL9205215 0.81 IDO1 (0.42) IDO1CDK2CCNA1CDK5CDK5R1
SCHEMBL9197120 0.73 ALOX5 (0.38) IDO1CDK5CDK5R1FFAR1ALDH1A1
SCHEMBL9200198 0.73 ALOX5 (0.38) IDO1CDK5CDK5R1FFAR1ALDH1A1
SCHEMBL9195547 0.71 IDO1 (0.43) IDO1CDK2CCNA1CDK5CDK5R1
SCHEMBL9852592 0.69 IDO1 (0.43) IDO1EPHX1HPGDSMN1; SMN2MAPT
SCHEMBL8604028 0.68 IDO1 (0.43) IDO1CDK2CCNA1CDK5CDK5R1
SCHEMBL8439880 0.68 IDO1 (0.43) IDO1CDK2CCNA1CDK5CDK5R1
SCHEMBL9206135 0.67 IDO1 (0.43) IDO1CDK2CCNA1CDK5CDK5R1
SCHEMBL9201296 0.67 CRBN (0.41) IDO1ALDH1A1HPGDSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0406863-B1 Cyclic amidinylthiocarbapenem derivatives BANYU PHARMA CO LTD (JP) 1995-05-24 EP disclosed
US-5100888-A Bactericides BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-03-31 US disclosed
EP-0406863-A1 Cyclic amidinylthiocarbapenem derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-01-09 EP disclosed