SCHEMBL9199449

SCHEMBL9199449

Cc1cc(NC(=O)CC#N)ccc1Br

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
KMT2A Q03164 4/20 0.59
RAB9A P51151 3/20 0.59
PKM P14618 1/20 0.59
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 2/20 0.57
MEN1 O00255 2/20 0.57
DRD4 P21917 2/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
MAPT P10636 3/20 0.53
RECQL P46063 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
LMNA P02545 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299426 0.88 CYP1A2 (0.57) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL11139407 0.86 CA12 (0.58) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL1259319 0.82 CYP1A2 (0.57) ALDH1A1KMT2ACYP1A2CYP2C19MEN1
SCHEMBL4003419 0.81 ALDH1A1 (0.69) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL848822 0.81 ALDH1A1 (0.69) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL11129650 0.81 KMT2A (0.70) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL13384768 0.80 CYP1A2 (0.58) ALDH1A1KMT2ACYP1A2CYP2C19MEN1
SCHEMBL11184694 0.80 CYP1A2 (0.58) ALDH1A1KMT2ACYP1A2CYP2C19MEN1
SCHEMBL7925078 0.80 ALDH1A1 (0.68) ALDH1A1KMT2ARAB9APKMCYP1A2
SCHEMBL19448886 0.80 PKM (0.68) ALDH1A1KMT2ARAB9APKMCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1030075-C 3-cycloalkyl-propionamides, their tautomers and their salts, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 1995-10-18 CN disclosed
EP-0484223-B1 3-Cycloalkylpropanamides, their tautomers and salts, process for their preparation, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1995-03-08 EP disclosed
US-5384423-A Intermediates for antiinflammatory agents ROUSSEL-UCLAF (FR) 1995-01-24 US disclosed
US-5308865-A Antiinflammatory agents ROUSSEL UCLAF (FR) 1994-05-03 US disclosed
US-5240960-A Antiinflammatory agents ROUSSEL UCLAF (FR) 1993-08-31 US disclosed
CN-1064482-A New 3-cycloalkyl-propanamides, the preparation method of their tautomer and its esters ROUSSEL UCLAF (FR) 1992-09-16 CN disclosed
EP-0484223-A2 3-Cycloalkylpropanamides, their tautomers and salts, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1992-05-06 EP disclosed
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed