SCHEMBL9200524

SCHEMBL9200524

O=C(O)c1cc(OCc2ccccc2)c(C(=O)c2ccccc2C(=O)OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
L3MBTL1 Q9Y468 4/20 0.52
CYP3A4 P08684 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
TDP1 Q9NUW8 3/20 0.50
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
HTT P42858 1/20 0.49
TSHR P16473 2/20 0.48
MAPK1 P28482 1/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A3 Q01959 1/20 0.48
POLB P06746 1/20 0.47
NR4A2 P43354 2/20 0.45
SRD5A2 P31213 1/20 0.45
NR4A1 P22736 1/20 0.44
NR4A3 Q92570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304467 0.89 ALDH1A1 (0.51) ALDH1A1NPSR1TDP1KMT2AMEN1
SCHEMBL9203039 0.88 ALDH1A1 (0.49) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL9195711 0.87 MEN1 (0.55) KMT2AMEN1HTTRAB9AFOLH1
SCHEMBL9203364 0.80 HTT (0.47) ALDH1A1L3MBTL1CYP3A4NPSR1CYP1A2
SCHEMBL9197479 0.80 MEN1 (0.56) KMT2AMEN1POLBNR4A2SRD5A2
SCHEMBL9195985 0.80 ALDH1A1 (0.55) ALDH1A1L3MBTL1CYP3A4NPSR1CYP1A2
SCHEMBL1316640 0.79 ALDH1A1 (0.56) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL9201021 0.78 PTGER1 (0.54) KMT2AMEN1HTTRAB9AFOLH1
SCHEMBL23809724 0.77 ALDH1A1 (0.62) ALDH1A1L3MBTL1CYP3A4NPSR1TDP1
SCHEMBL3634188 0.77 ALDH1A1 (0.80) ALDH1A1L3MBTL1CYP3A4NPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687249-A1 BALANOIDS ELI LILLY AND COMPANY (US) 1995-12-20 EP disclosed
WO-1994020062-A2 BALANOIDS AS PROTEIN KINASE C INHIBITORS ELI LILLY AND COMPANY (US) 1994-09-15 WO disclosed