SCHEMBL9200650

SCHEMBL9200650

Cc1ccc(N2CCC(CCO)C2)nn1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.40
P2RX7 Q99572 1/20 0.39
MAPT P10636 1/20 0.39
PIK3CA P42336 2/20 0.38
MTOR P42345 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PTGER4 P35408 1/20 0.37
GLS O94925 5/20 0.37
PDE10A Q9Y233 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9195135 0.93 MAP4K4 (0.40) NR1I2P2RX7MAPTPIK3CAMTOR
SCHEMBL1562375 0.91 MAPT (0.43) MAPTPIK3CAMTORMEN1KMT2A
SCHEMBL18291297 0.88 PTGER4 (0.46) NR1I2PIK3CAMTORPTGER4GLS
SCHEMBL9200293 0.85 NR1I2 (0.40) NR1I2MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL9197797 0.82 CYP11B2 (0.48) NR1I2MAPTPIK3CAMTORMEN1
SCHEMBL9195108 0.81 PDE10A (0.44) NR1I2PIK3CAMTORMEN1KMT2A
SCHEMBL2146739 0.80 PDE10A (0.56) MAPTPIK3CAMTORIRAK4PDE10A
SCHEMBL2146743 0.80 PDE10A (0.56) MAPTPIK3CAMTORIRAK4PDE10A
SCHEMBL2146811 0.80 PDE10A (0.56) MAPTPIK3CAMTORIRAK4PDE10A
SCHEMBL18291295 0.80 NR1I2 (0.46) NR1I2KMT2APTGER4PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0435381-B1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA NV (BE) 1995-11-02 EP disclosed
US-5196535-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-23 US disclosed
US-5100893-A Viricides, effective against picorna virus, durability JANSSEN PHARMACEUTICA N.V. (BE) 1992-03-31 US disclosed
EP-0435381-A1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-07-03 EP disclosed