SCHEMBL9200670

SCHEMBL9200670

Cc1ccc(C(=O)NC2CCC(CCN3CCN(c4ccccn4)CC3)CC2)cc1

nearest known ligand 0.85

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.85
DRD3 P35462 15/20 0.69
HTR2A P28223 10/20 0.56
ALDH1A1 P00352 2/20 0.55
HTR1A P08908 2/20 0.54
DRD4 P21917 1/20 0.52
HTR2C P28335 1/20 0.52
HTR2B P41595 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199135 0.92 DRD2 (1.00) DRD2DRD3HTR2AALDH1A1HTR1A
SCHEMBL9196530 0.90 DRD2 (0.85) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL9841829 0.90 DRD2 (0.81) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL9197525 0.90 DRD2 (0.81) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL9197530 0.90 DRD2 (0.81) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL9196198 0.86 DRD2 (0.78) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL9197591 0.86 DRD2 (0.77) DRD2DRD3HTR2AALDH1A1HTR1A
SCHEMBL13415659 0.86 DRD2 (0.77) DRD2DRD3HTR2AALDH1A1HTR1A
SCHEMBL9202518 0.85 DRD2 (0.79) DRD2DRD3HTR2AALDH1A1HTR1A
SCHEMBL9202507 0.85 DRD2 (0.79) DRD2DRD3HTR2AALDH1A1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed