SCHEMBL9200941

SCHEMBL9200941

OC1(c2cccnc2)CCC(CCN2CC=C(c3ccccc3)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.54
DRD3 P35462 5/20 0.54
DRD4 P21917 4/20 0.51
SIGMAR1 Q99720 2/20 0.45
CCR1 P32246 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200937 1.00 DRD2 (0.54) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9200935 1.00 DRD2 (0.54) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9200032 0.82 DRD2 (0.60) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9200022 0.82 DRD2 (0.60) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9202901 0.82 DRD2 (0.60) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9199080 0.80 ALDH1A1 (0.47) MEN1KMT2AALDH1A1LMNA
SCHEMBL9199075 0.80 ALDH1A1 (0.47) MEN1KMT2AALDH1A1LMNA
SCHEMBL9199068 0.80 ALDH1A1 (0.47) MEN1KMT2AALDH1A1LMNA
SCHEMBL9196981 0.78 DRD2 (0.53) DRD2DRD3DRD4SIGMAR1CCR1
SCHEMBL9196980 0.78 DRD2 (0.53) DRD2DRD3DRD4SIGMAR1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed