SCHEMBL9201002

SCHEMBL9201002

CCCC(c1ccncc1F)n1ccc2cc(OCc3ccccc3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.43
ROCK1 Q13464 1/20 0.43
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP26A1 O43174 1/20 0.37
CYP3A4 P08684 1/20 0.37
SRD5A2 P31213 1/20 0.37
ALOX5 P09917 1/20 0.37
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
GRM2 Q14416 2/20 0.35
GPR132 Q9UNW8 3/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9194455 0.84 SLC6A2 (0.63) SLC6A2ROCK1MEN1NPC1RAB9A
SCHEMBL9500230 0.84 BCHE (0.43) MEN1NPC1RAB9AKMT2AGRM2
SCHEMBL9194863 0.81 SLC6A2 (0.65) SLC6A2
Oxalic Acid SCHEMBL9196754 0.80 SLC6A2 (0.57) SLC6A2ROCK1MEN1NPC1RAB9A
SCHEMBL9739947 0.80 ROCK1 (0.43) ROCK1MEN1NPC1RAB9AKMT2A
SCHEMBL8845681 0.79 BCHE (0.48) SLC6A2
Hydrochloric Acid SCHEMBL8544423 0.79 ROCK1 (0.42) ROCK1MEN1NPC1RAB9AKMT2A
SCHEMBL14977575 0.79 NPC1 (0.50) ROCK1MEN1NPC1RAB9AKMT2A
SCHEMBL8845692 0.78 BCHE (0.41) SLC6A2
SCHEMBL7621050 0.74 BCHE (0.51) SLC6A2ROCK1MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US claimed
EP-0471296-B1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST ROUSSEL PHARMA (US) 1995-11-08 EP disclosed
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0471296-A1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed