SCHEMBL9201214

SCHEMBL9201214

Cc1coc(C)c1C(=O)Nc1ccc(Cl)c(C(=O)OC(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
LMNA P02545 7/20 0.43
KMT2A Q03164 5/20 0.43
MAPT P10636 5/20 0.43
MEN1 O00255 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 2/20 0.43
RXFP1 Q9HBX9 1/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
HTR1E P28566 2/20 0.41
S1PR3 Q99500 2/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CSF1R P07333 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27312850 0.84 NPC1 (0.60) NPC1RAB9AMAPTSMN1; SMN2KDM4E
SCHEMBL9199855 0.83 KMT2A (0.50) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL9205677 0.81 SMN1; SMN2 (0.57) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL9203674 0.81 GRM1 (0.53) NPC1RAB9AKMT2AMAPTMEN1
SCHEMBL9199828 0.79 AKR1C3 (0.56) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL8930039 0.79 DHODH (0.56) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL9201230 0.78 MAPT (0.48) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL8929781 0.78 HPGD (0.58) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL27309634 0.77 RAB9A (0.66) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL6362855 0.76 LMNA (0.50) NPC1RAB9ALMNAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497816-B1 TREATMENT OF HIV INFECTIONS AND COMPOUNDS USEFUL THEREIN UNIROYAL CHEMICAL LTD (CA) 1995-05-17 EP claimed
EP-0497816-A1 TREATMENT OF HIV INFECTIONS AND COMPOUNDS USEFUL THEREIN. UNIROYAL CHEMICAL LTD (CA) 1992-08-12 EP claimed
WO-1991005761-A1 TREATMENT OF HIV INFECTIONS AND COMPOUNDS USEFUL THEREIN UNIROYAL CHEMICAL LTD./UNIROYAL CHEMICAL LTEE (CA) 1991-05-02 WO claimed