SCHEMBL9201249

SCHEMBL9201249

CC(C)c1ccc(C2(Cn3cncn3)OCC2(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 2/20 0.37
CYP19A1 P11511 1/20 0.36
CYP3A4 P08684 8/20 0.35
THRB P10828 1/20 0.35
CYP2C9 P11712 5/20 0.34
CYP1A2 P05177 4/20 0.34
CYP2C19 P33261 4/20 0.34
CYP2D6 P10635 3/20 0.34
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201238 0.88 CYP3A4 (0.46) HSP90AA1NPSR1CYP3A4THRBCYP2C9
SCHEMBL9203098 0.86 HSP90AA1 (0.51) HSP90AA1NPSR1MAPTCYP19A1CYP3A4
SCHEMBL9198433 0.85 CYP3A4 (0.45) HSP90AA1NPSR1CYP19A1CYP3A4THRB
SCHEMBL9201064 0.83 ALDH1A1 (0.50) HSP90AA1NPSR1MAPTCYP19A1CYP3A4
SCHEMBL9201132 0.80 HSP90AA1 (0.38) HSP90AA1NPSR1MAPTCYP19A1CYP3A4
SCHEMBL9195001 0.78 HSP90AA1 (0.40) HSP90AA1NPSR1MAPTCYP19A1CYP3A4
SCHEMBL10594715 0.75 HSP90AA1 (0.36) HSP90AA1NPSR1MAPTCYP19A1CYP3A4
SCHEMBL9202244 0.74 CYP3A4 (0.58) HSP90AA1MAPTCYP3A4THRBCYP2C9
SCHEMBL9200532 0.71 CYP3A4 (0.42) HSP90AA1CYP19A1CYP3A4THRBCYP2C9
SCHEMBL9314674 0.71 CYP3A4 (0.44) HSP90AA1NPSR1MAPTCYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431968-B1 Oxetane derivatives, their preparation and their use as anti-fungal or fungicidal agents SANKYO CO (JP) 1995-03-15 EP disclosed
US-5134152-A 1,2,4-Triazole compounds SANKYO COMPANY, LIMITED (JP) 1992-07-28 US disclosed
EP-0431968-A1 Oxetane derivatives, their preparation and their use as anti-fungal or fungicidal agents Sankyo Company Limited (JP) 1991-06-12 EP disclosed