SCHEMBL9201517

SCHEMBL9201517

CCCCCCc1cn[c]s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 3/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK5 Q00535 1/20 0.34
PTGS2 P35354 3/20 0.33
ESR1 P03372 2/20 0.33
ADRA2A P08913 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
TACR2 P21452 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
LMNA P02545 1/20 0.33
SHBG P04278 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5004070 0.92
SCHEMBL987593 0.67 ESR1 (0.38) KCNH2ALDH1A1PTGS2ESR1ADRA2A
SCHEMBL1286045 0.67 ESR1 (0.38) KCNH2ALDH1A1PTGS2ESR1ADRA2A
SCHEMBL735087 0.67 ESR1 (0.38) KCNH2ALDH1A1PTGS2ESR1ADRA2A
SCHEMBL1285757 0.67 ESR1 (0.38) KCNH2ALDH1A1PTGS2ESR1ADRA2A
SCHEMBL16892538 0.67 ESR1 (0.38) KCNH2ALDH1A1PTGS2ESR1ADRA2A
SCHEMBL19861696 0.67 TBXAS1 (0.39) KCNH2ALDH1A1TDP1L3MBTL1PTGS2
SCHEMBL16266833 0.67 TBXAS1 (0.39) KCNH2ALDH1A1TDP1L3MBTL1PTGS2
SCHEMBL21230535 0.67 KCNH2 (0.38) KCNH2ALDH1A1TDP1L3MBTL1PTGS2
SCHEMBL8923831 0.66 ESR1 (0.45) KCNH2ALDH1A1PTGS2ESR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214476-B One class contains 4-methyl isophthalic acid, carboxamidine derivatives of 2,3-thiadiazoles and its production and use NANKAI UNIVERSITY (CN) 2016-03-02 CN claimed
CN-103214476-A Formamidine derivatives containing 4-methyl-1,2,3-thiadiazole, and preparation methods and uses UNIV NANKAI 2013-07-24 CN claimed
CN-103214476-B One class contains 4-methyl isophthalic acid, carboxamidine derivatives of 2,3-thiadiazoles and its production and use NANKAI UNIVERSITY (CN) 2016-03-02 CN disclosed
CN-103214476-A Formamidine derivatives containing 4-methyl-1,2,3-thiadiazole, and preparation methods and uses UNIV NANKAI 2013-07-24 CN disclosed
CN-1029227-C Composition for denatured denaturation or protection agent for nerve cell and process for preparing benzene derivatives used for composition OTSUKA PHARMA CO LTD (JP) 1995-07-05 CN disclosed
EP-0382213-B1 Biphenyl derivative, nerve cell degeneration repairing or protecting agent and process for preparing a phenyl derivative contained in the agent OTSUKA PHARMA CO LTD (JP) 1995-05-10 EP disclosed
US-5053548-A Containing hydroxy substituents; nervous system disorders OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1991-10-01 US disclosed
CN-1044807-A Neurocyte sex change reparation or protective material are with composition and the preparation method that is used for the benzene derivative of said composition OTSUKA PHARMA CO LTD (JP) 1990-08-22 CN disclosed
EP-0382213-A2 Biphenyl derivative, nerve cell degeneration repairing or protecting agent and process for preparing a phenyl derivative contained in the agent OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed