SCHEMBL9201549

SCHEMBL9201549

CS(=O)(=O)c1ccc(-n2nc(C#N)cc2-c2ccc(F)cc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.78
PTGS1 P23219 5/20 0.67
AOC3 Q16853 1/20 0.60
CYP2C9 P11712 1/20 0.54
ALOX5 P09917 1/20 0.52
NR3C2 P08235 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203156 1.00 PTGS2 (0.78) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL9203630 0.89 PTGS2 (0.65) PTGS2PTGS1CYP2C9ALOX5
SCHEMBL7459996 0.89 PTGS2 (0.62) PTGS2PTGS1CYP2C9ALOX5
SCHEMBL9207728 0.88 PTGS2 (0.64) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL215235 0.88 PTGS2 (1.00) PTGS2PTGS1CYP2C9
SCHEMBL27342072 0.88 ALOX5 (0.61) PTGS2PTGS1CYP2C9ALOX5
SCHEMBL9210297 0.87 PTGS2 (0.60) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL9210069 0.87 PTGS2 (0.60) PTGS2PTGS1ALOX5
SCHEMBL9209500 0.86 PTGS2 (0.59) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL7878979 0.86 PTGS2 (0.59) PTGS2PTGS1AOC3CYP2C9ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1046506-C Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-11-17 CN disclosed
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
US-5134142-A PYRAZOLE DERIVATIVES, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-07-28 US disclosed
CN-1050382-A Pyrazole derivatives and preparation method thereof and medicinal compositions FUJISAWA PHARMACEUTICAL CO (JP) 1991-04-03 CN disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed