SCHEMBL9201743

SCHEMBL9201743

CS(=O)(=O)c1ccc(-c2cc(N)nn2-c2ccc(F)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.71
PTGS1 P23219 4/20 0.71
AOC3 Q16853 1/20 0.64
CYP2C9 P11712 1/20 0.57
ALOX5 P09917 1/20 0.55
CHRNA7 P36544 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15463064 0.86 ALOX5 (0.73) PTGS2PTGS1CYP2C9ALOX5
SCHEMBL8421061 0.85 PTGS2 (0.88) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL9203342 0.85 PTGS2 (0.73) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL14280456 0.85 ALOX5 (0.76) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL9207256 0.84 PTGS2 (0.71) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL28740979 0.84 PTGS2 (0.71) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL9210255 0.84 PTGS2 (0.67) PTGS2PTGS1AOC3CYP2C9ALOX5
SCHEMBL5229949 0.83 PTGS2 (1.00) PTGS2PTGS1CYP2C9ALOX5
Sc-58125 SCHEMBL12375146 0.83 PTGS2 (1.00) PTGS2PTGS1CYP2C9ALOX5
Sc-58125 SCHEMBL214120 0.83 PTGS2 (1.00) PTGS2PTGS1CYP2C9ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
US-5134142-A PYRAZOLE DERIVATIVES, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-07-28 US disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed