SCHEMBL9203069

SCHEMBL9203069

NCC(c1ccccc1)n1ccc2cccnc21

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.43
P2RX7 Q99572 1/20 0.43
CYP2C19 P33261 1/20 0.41
PARP1 P09874 1/20 0.41
SLC6A2 P23975 3/20 0.39
CDC7 O00311 1/20 0.38
CDK2 P24941 1/20 0.38
ENPP1 P22413 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HTR2A P28223 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
MTNR1A P48039 1/20 0.35
SLC22A12 Q96S37 1/20 0.34
RPS6KB1 P23443 1/20 0.34
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3229386 0.83 SLC6A2 (0.43) SLC6A4P2RX7CYP2C19PARP1SLC6A2
SCHEMBL3226894 0.80 SLC6A2 (0.66) SLC6A4P2RX7SLC6A2HTR2AMTNR1A
SCHEMBL9206196 0.80 CYP2C19 (0.40) SLC6A4P2RX7CYP2C19PARP1SLC6A2
SCHEMBL2586507 0.80 P2RX7 (0.50) P2RX7CYP2C19PARP1CDC7CDK2
SCHEMBL4087126 0.73 SLC6A4 (0.49) SLC6A4P2RX7CYP2C19PARP1SLC6A2
SCHEMBL9266746 0.73 PARP1 (0.39) SLC6A4P2RX7CYP2C19PARP1SLC6A2
SCHEMBL8135638 0.71 PARP1 (0.47) CYP2C19PARP1CDC7CDK2HTR2A
SCHEMBL23938013 0.71 PARP1 (0.46) CYP2C19PARP1CDC7CDK2ENPP1
SCHEMBL598048 0.71 PARP1 (0.46) CYP2C19PARP1CDC7CDK2ENPP1
SCHEMBL30991276 0.71 PARP1 (0.46) CYP2C19PARP1CDC7CDK2ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557171-B1 Azaindoles, process for their preparation and medicines containing them LIPHA (FR) 1995-07-19 EP disclosed
US-5338849-A Treating hyperlipidemia, atherosclerosis LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1994-08-16 US disclosed
EP-0557171-A1 Azaindoles, process for their preparation and medicines containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1993-08-25 EP disclosed