SCHEMBL9206196

SCHEMBL9206196

O=[N+]([O-])CC(c1ccccc1)n1ccc2cccnc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
CNR1 P21554 3/20 0.40
P2RX7 Q99572 1/20 0.39
PARP1 P09874 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
NPC1 O15118 2/20 0.36
ADAM17 P78536 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 2/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ENPP1 P22413 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203069 0.80 SLC6A4 (0.43) CYP2C19P2RX7PARP1SLC22A12KDM4E
SCHEMBL3229386 0.77 SLC6A2 (0.43) CYP2C19P2RX7PARP1SLC22A12KDM4E
SCHEMBL3226894 0.74 SLC6A2 (0.66) P2RX7SLC6A2SLC6A4MTNR1A
SCHEMBL2586507 0.74 P2RX7 (0.50) CYP2C19P2RX7PARP1SLC22A12KDM4E
SCHEMBL27984061 0.70 NPC1 (0.41) CNR1NPC1ADAM17KDM4EMAPT
SCHEMBL4087126 0.68 SLC6A4 (0.49) CYP2C19P2RX7PARP1SLC6A2SLC6A4
SCHEMBL9266746 0.68 PARP1 (0.39) CYP2C19P2RX7PARP1SLC22A12MAPT
SCHEMBL28041794 0.68 ALDH1A1 (0.48) CNR1KDM4EMAPTPKMALDH1A1
SCHEMBL20181945 0.67 PARP1 (0.41) CYP2C19P2RX7PARP1SLC22A12SLC6A2
SCHEMBL28137577 0.67 CNR1 (0.43) CNR1KDM4EMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557171-B1 Azaindoles, process for their preparation and medicines containing them LIPHA (FR) 1995-07-19 EP disclosed
US-5338849-A Treating hyperlipidemia, atherosclerosis LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1994-08-16 US disclosed
EP-0557171-A1 Azaindoles, process for their preparation and medicines containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1993-08-25 EP disclosed