SCHEMBL9203280

SCHEMBL9203280

NC(Cc1ccccc1)C(=O)N(Cc1ccc(O)cc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.50
ALPI P09923 1/20 0.45
PKM P14618 1/20 0.45
PTGS1 P23219 1/20 0.45
XIAP P98170 1/20 0.45
MC4R P32245 4/20 0.45
MC5R P33032 3/20 0.45
MC3R P41968 3/20 0.45
TDP1 Q9NUW8 1/20 0.44
HDAC8 Q9BY41 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SLC15A1 P46059 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
BACE1 P56817 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388851 0.90 SLC7A5 (0.43) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL9200732 0.86 DPP7 (0.41) SLC7A5MC4RMC5RMC3RTDP1
SCHEMBL9198257 0.84 TDP1 (0.49) SLC7A5TDP1MEN1KMT2AOPRD1
SCHEMBL9198245 0.84 TDP1 (0.49) SLC7A5TDP1MEN1KMT2AOPRD1
SCHEMBL9195704 0.82 ALDH1A1 (0.39) MC4RTDP1MEN1KMT2A
SCHEMBL9203137 0.80 TDP1 (0.46) TDP1MEN1KMT2A
SCHEMBL9196505 0.80 TDP1 (0.50) SLC7A5TDP1MEN1KMT2A
SCHEMBL8119790 0.76 EPHX1 (0.44) SLC7A5TDP1MEN1KMT2AOPRD1
SCHEMBL4156779 0.75 OPRM1 (0.53) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL29053326 0.74 SLC7A5 (0.50) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed