SCHEMBL9205183

SCHEMBL9205183

C=CCc1cccc(C=C(OCC)C(=O)c2ccc(C(=O)N(C)C)cc2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PTGS2 P35354 1/20 0.34
ALDH1A1 P00352 6/20 0.34
KDM4E B2RXH2 3/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
CYP1A2 P05177 2/20 0.33
TSHR P16473 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208251 0.92 PRSS1 (0.33) CYP3A4MEN1KMT2ATDP1L3MBTL1
SCHEMBL9197566 0.90 MAPT (0.35) CYP3A4MEN1KMT2AALDH1A1HPGD
SCHEMBL9204247 0.89 CYP3A4 (0.37) CYP3A4MEN1KMT2ATDP1L3MBTL1
SCHEMBL9203046 0.87 CYP4F2 (0.38) CYP3A4MEN1KMT2ATDP1ALDH1A1
SCHEMBL9206935 0.86 SLC7A5 (0.35) CYP3A4MEN1KMT2ATDP1L3MBTL1
SCHEMBL9206870 0.86 PTGS2 (0.38) CYP3A4MEN1KMT2ATDP1L3MBTL1
SCHEMBL9206999 0.84 HPGD (0.40) CYP3A4MEN1KMT2ATDP1L3MBTL1
SCHEMBL9203895 0.81 MEN1 (0.51) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL9198798 0.80 HDAC8 (0.40) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL9206588 0.79 CYP11B1 (0.34) CYP3A4KMT2AALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed