SCHEMBL9207618

SCHEMBL9207618

COc1cc2c(cc1OC)CN(CC1CCN(CCc3cccc(C)n3)C1)CC2

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.47
BCHE P06276 1/20 0.47
HTR7 P34969 1/20 0.45
ADRA1B P35368 1/20 0.44
ABCB1 P08183 7/20 0.43
ABCC1 P33527 1/20 0.43
DHCR7 Q9UBM7 2/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217614 0.94 ACHE (0.50) ACHEBCHEHTR7ADRA1BABCB1
SCHEMBL9214063 0.88 BCHE (0.44) ACHEBCHEHTR7ADRA1BABCB1
SCHEMBL9210290 0.85 KCNH2 (0.41) ACHEBCHE
SCHEMBL9204663 0.83 ACHE (0.52) ACHEBCHEADRA1B
SCHEMBL9212638 0.82 ACHE (0.53) ACHEBCHEADRA1B
SCHEMBL9204444 0.80 KDM4E (0.43) ACHEBCHE
Hydrochloric Acid SCHEMBL9206759 0.79 DHCR7 (0.64) ABCB1DHCR7
Hydrochloric Acid SCHEMBL9215875 0.79 ABCB1 (0.54) ABCB1DHCR7
SCHEMBL9206874 0.79 BCHE (0.42) ACHEBCHEADRA1B
Hydrochloric Acid SCHEMBL9740423 0.79 CYP3A4 (0.42) ACHEBCHEADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed