SCHEMBL9210290

SCHEMBL9210290

Cc1cccc(CCN2CCC(CN3CCc4cc(C)c(C)cc4CC3)C2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 2/20 0.40
POLB P06746 1/20 0.40
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
PDE2A O00408 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GNRHR P30968 1/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9206993 0.86 KCNH2 (0.38) KCNH2CYP2D6CYP3A4CYP2C19KDM4E
SCHEMBL9207618 0.85 ACHE (0.47) BCHEACHE
SCHEMBL9217614 0.80 ACHE (0.50) KCNH2CYP2D6CYP3A4CYP2C19KDM4E
SCHEMBL9204444 0.79 KDM4E (0.43) KCNH2CYP2D6CYP3A4CYP2C19KDM4E
SCHEMBL9209361 0.79 KCNH2 (0.46) KCNH2CYP2D6CYP3A4CYP2C19KDM4E
SCHEMBL9216817 0.78 BCHE (0.38) KCNH2CYP2D6CYP3A4CYP2C19KDM4E
SCHEMBL9204663 0.76 ACHE (0.52) BCHEACHEMEN1KMT2A
SCHEMBL9211917 0.75 HTR1A (0.46) ACHEMEN1KMT2ASIGMAR1
SCHEMBL9210283 0.75 SIGMAR1 (0.42) SIGMAR1HRH1HRH3
SCHEMBL9214063 0.74 BCHE (0.44) KDM4EBCHEACHELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed