SCHEMBL9207791

SCHEMBL9207791

FC(F)(F)c1cccc(N2CCN(CCCCc3c[nH]c4ccccc34)CC2)n1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 14/20 0.60
DRD2 P14416 5/20 0.54
HTR2A P28223 3/20 0.53
HTR7 P34969 3/20 0.53
HTR6 P50406 2/20 0.53
SLC6A4 P31645 1/20 0.51
HRH1 P35367 1/20 0.51
DRD3 P35462 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207116 0.97 HTR1A (0.63) HTR1ADRD2
SCHEMBL9205998 0.93 HTR2A (0.56) HTR1ADRD2HTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL9207142 0.92 HTR2A (0.55) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL9206679 0.85 HTR1A (0.63) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL9211981 0.81 HTR1A (0.67) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL9207621 0.81 HTR1A (0.64) HTR1AHTR7HTR6SLC6A4
Hydrochloric Acid SCHEMBL9213499 0.81 HTR1A (0.66) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL9205636 0.80 HTR1A (0.54) HTR1ADRD2HTR7HTR6
SCHEMBL9206516 0.78 HTR2A (0.60) HTR1ADRD2HTR2A
SCHEMBL9207839 0.77 HTR1A (0.61) HTR1ADRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP claimed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US claimed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP claimed