SCHEMBL9208573

SCHEMBL9208573

COc1cccc(CCCN2CCCC(CN3Cc4cc(OC)c(OC)cc4C3=O)C2)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
CHRNB2 P17787 2/20 0.47
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
CHRNA4 P43681 2/20 0.47
HTR2A P28223 2/20 0.44
SIGMAR1 Q99720 1/20 0.44
CCR3 P51677 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
ACHE P22303 1/20 0.43
ABCB1 P08183 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9214816 0.94 MEN1 (0.53) MEN1KMT2ASIGMAR1HRH3
SCHEMBL9216672 0.91 CHRNB2 (0.47) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL9207276 0.90 ABCB1 (0.47) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL9207682 0.88 CHRNB2 (0.45) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL9212297 0.86 CHRNB4 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4ABCB1
SCHEMBL9211577 0.86 BCHE (0.46) MEN1KMT2ACHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL9210506 0.85 CHRNB4 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9212603 0.85 GAA (0.50) MEN1KMT2AHRH3ABCB1
Hydrochloric Acid SCHEMBL9214061 0.85 MEN1 (0.46) MEN1KMT2AABCB1
Hydrochloric Acid SCHEMBL9210830 0.82 CHRNB2 (0.46) MEN1KMT2ACHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed