SCHEMBL9216672

SCHEMBL9216672

COc1ccc(CCCN2CCCC(CN3Cc4cc(OC)c(OC)cc4C3=O)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.47
CHRNB4 P30926 3/20 0.47
CHRNA3 P32297 3/20 0.47
CHRNA4 P43681 3/20 0.47
GAA P10253 1/20 0.45
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
ABCB1 P08183 1/20 0.41
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207682 0.97 CHRNB2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4GAA
SCHEMBL9212603 0.95 GAA (0.50) GAAMEN1KMT2ANPC1RAB9A
SCHEMBL9212297 0.92 CHRNB4 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4ABCB1
SCHEMBL9207276 0.92 ABCB1 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4GAA
Hydrochloric Acid SCHEMBL9210830 0.91 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4GAA
SCHEMBL9208573 0.91 MEN1 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4MEN1
SCHEMBL9216056 0.87 BCHE (0.44) CHRNB2CHRNB4CHRNA3CHRNA4GAA
Hydrochloric Acid SCHEMBL9214061 0.87 MEN1 (0.46) GAAMEN1KMT2ANPC1RAB9A
Hydrochloric Acid SCHEMBL9208088 0.87 ABCB1 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4ABCB1
SCHEMBL9212017 0.86 GAA (0.46) CHRNB2CHRNB4CHRNA3CHRNA4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed