SCHEMBL9209352

SCHEMBL9209352

CC(=O)NCCNc1nnc(NCCNC(C)=O)c2cc3ccccc3cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA4 P22748 1/20 0.56
CA7 P43166 1/20 0.56
CA9 Q16790 1/20 0.56
CA14 Q9ULX7 1/20 0.56
CYP1A2 P05177 14/20 0.50
CYP3A4 P08684 12/20 0.50
CYP2D6 P10635 11/20 0.50
CLK4 Q9HAZ1 8/20 0.50
ALDH1A1 P00352 7/20 0.50
TSHR P16473 6/20 0.50
CYP2C19 P33261 5/20 0.50
HSD17B10 Q99714 4/20 0.50
CYP2C9 P11712 2/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ALOX15 P16050 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421485 0.77 SOD1 (0.51) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL9201354 0.75 SOD1 (0.47) ALDH1A1CYP2C19KDM4ELMNAMAPT
SCHEMBL9209228 0.75 CYP1A2 (0.51) CA12CA4CA7CA9CA14
SCHEMBL9208673 0.74 SOD1 (0.56) ALDH1A1TSHRHSD17B10MEN1KMT2A
SCHEMBL8421424 0.74 SOD1 (0.56) CYP3A4CYP2D6ALDH1A1KDM4ELMNA
SCHEMBL8423745 0.73 SOD1 (0.47) CYP1A2MEN1KMT2AKDM4EADORA2A
SCHEMBL9204316 0.73 TOP2A (0.52) MEN1KMT2A
Hydrochloric Acid SCHEMBL8421903 0.73 SOD1 (0.55) CYP3A4CYP2D6ALDH1A1KDM4ELMNA
SCHEMBL11882576 0.72 CA12 (1.00) CA12CA4CA7CA9CA14
SCHEMBL9202631 0.72 TOP2A (0.45) CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497809-B1 1,4-BIS(ALKYLAMINO)-2,3-DIAZA-ANTHRACENE-9,10-DIONES BOEHRINGER MANNHEIM ITALIA (IT) 1995-06-28 EP disclosed
US-5162320-A 1,4-BIS(ALKYLAMINO)-2,3-DIAZA-ANTHRACENE-9,10-DIONES BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1992-11-10 US disclosed
EP-0497809-A1 1,4-BIS(ALKYLAMINO)-2,3-DIAZA-ANTHRACENE-9,10-DIONES. BOEHRINGER MANNHEIM ITALIA (IT) 1992-08-12 EP disclosed
WO-1991006540-A1 1,4-BIS(ALKYLAMINO)-2,3-DIAZA-ANTHRACENE-9,10-DIONES BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1991-05-16 WO disclosed