SCHEMBL9210237

SCHEMBL9210237

Cc1cc(CCCCCOc2c(Cl)cc(-c3nc(C)no3)cc2Cl)on1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
ACHE P22303 2/20 0.39
BCHE P06276 1/20 0.39
LRRK2 Q5S007 2/20 0.38
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
IGF1R P08069 2/20 0.32
FGFR1 P11362 2/20 0.32
KDR P35968 2/20 0.32
SCARB1 Q8WTV0 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
INSR P06213 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201847 0.88 NR1I2 (0.56) NR1I2CYP3A4CYP2D6ACHEBCHE
SCHEMBL9705958 0.85 NR1I2 (0.42) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9705948 0.84 NR1I2 (0.43) NR1I2CYP3A4CYP2D6MAPTMEN1
SCHEMBL9207573 0.84 NR1I2 (0.41) NR1I2CYP3A4CYP2D6LRRK2MAPT
SCHEMBL9705774 0.84 NR1I2 (0.41) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9200228 0.83 NR1I2 (0.40) NR1I2CYP3A4CYP2D6MAPTMEN1
SCHEMBL9204655 0.83 NR1I2 (0.61) NR1I2CYP3A4CYP2D6ACHEBCHE
SCHEMBL9210194 0.83 NR1I2 (0.53) NR1I2CYP3A4CYP2D6MAPTMEN1
SCHEMBL9436214 0.82 NR1I2 (0.43) NR1I2CYP3A4CYP2D6MAPTMEN1
SCHEMBL9436119 0.81 PTGS2 (0.40) NR1I2CYP3A4CYP2D6TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413289-B1 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC (US) 1995-02-01 EP disclosed
US-5175178-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING DRUG INC. (US) 1992-12-29 US disclosed
EP-0413289-A2 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1991-02-20 EP disclosed
US-4942241-A PICORNAVIRUS INCLUDING RHINOVIRUS STERLING DRUG INC. (US) 1990-07-17 US disclosed