SCHEMBL9210499

SCHEMBL9210499

COc1ccc2[nH]cc(CCCN3CCC(CN4Cc5cc6c(cc5C4)OCO6)C3)c2c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.59
SLC6A2 P23975 3/20 0.53
SLC6A4 P31645 3/20 0.53
SLC6A3 Q01959 3/20 0.53
DRD2 P14416 1/20 0.51
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
ADRA1D P25100 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
HTR2A P28223 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213471 0.83 HTR1A (0.61) HTR1ASLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL9214106 0.83 HTR1A (0.61) HTR1ASLC6A2SLC6A4SLC6A3ADRA2A
SCHEMBL9210128 0.82 HTR1A (0.45) HTR1ASLC6A2SLC6A4SLC6A3DRD2
SCHEMBL8555361 0.78 HTR1A (0.65) HTR1ASLC6A4DRD2ADRA2AADRA2B
Hydrochloric Acid SCHEMBL9207604 0.78 HTR1A (0.52) HTR1ASLC6A2SLC6A4SLC6A3DRD2
SCHEMBL9206604 0.78 HTR1A (0.55) HTR1ASLC6A2SLC6A4SLC6A3ADRA2A
Hydrochloric Acid SCHEMBL9743101 0.77 HTR1A (0.52) HTR1ASLC6A4SLC6A3DRD2HTR2A
SCHEMBL9209371 0.77 HTR1D (0.52) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL9206815 0.77 HTR1A (0.55) HTR1ASLC6A4DRD2HTR2A
SCHEMBL8871000 0.76 HTR1A (0.62) HTR1ADRD2ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed