SCHEMBL9210508

SCHEMBL9210508

Cc1cc2c(cc1C)CC(=O)N(CC1CCCN(CCCc3cccnc3)C1)C=C2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.37
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
CHRNB4 P30926 5/20 0.35
CHRNA3 P32297 5/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CHRNB2 P17787 3/20 0.35
CHRNA4 P43681 3/20 0.35
KAT2B Q92831 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9741720 0.98 CCR2 (0.36) CCR2KCNH2HRH3CHRNB4CHRNA3
SCHEMBL9739274 0.90 CHRNB4 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL9213548 0.88 PDE5A (0.37) CCR2KCNH2HRH3CHRNB4CHRNA3
SCHEMBL9214964 0.88 CHRNB4 (0.41) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL9215863 0.85 BRD4 (0.40) CHRNB4CHRNA3CHRM2CHRM1CHRM3
SCHEMBL9213488 0.83 NAMPT (0.39) CCR2KCNH2HRH3CHRNB4CHRNA3
SCHEMBL9212245 0.82 CHRNB4 (0.43) CHRNB4CHRNA3CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL9740467 0.82 NAMPT (0.38) CCR2KCNH2HRH3CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL9739435 0.81 CHRNB4 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL9740211 0.80 HRH3 (0.43) CCR2KCNH2HRH3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed