SCHEMBL9212245

SCHEMBL9212245

COc1cc2c(cc1OC)CC(=O)N(CCCC1CCCN(CCCc3cccnc3)C1)C=C2

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 4/20 0.43
CHRNA3 P32297 4/20 0.43
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
PDE4D Q08499 1/20 0.39
HCN4 Q9Y3Q4 3/20 0.38
BRD4 O60885 1/20 0.38
PTAFR P25105 6/20 0.38
HTR2A P28223 1/20 0.37
FKBP1A P62942 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9739435 0.98 CHRNB4 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
SCHEMBL9739274 0.92 CHRNB4 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
SCHEMBL9214964 0.90 CHRNB4 (0.41) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
SCHEMBL9215863 0.88 BRD4 (0.40) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
Hydrochloric Acid SCHEMBL9739444 0.83 CYP3A4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
SCHEMBL9210508 0.82 CCR2 (0.37) CHRNB4CHRNA3CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL9741720 0.81 CCR2 (0.36) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL9209351 0.81 CHRNB4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
Hydrochloric Acid SCHEMBL9740808 0.80 CHRNB4 (0.45) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D
Hydrochloric Acid SCHEMBL10649892 0.79 CHRNB4 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed